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(-)-Bicuculline methochloride
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Catalog No. T12044Cas No. 53552-05-9
Alias l-Bicuculline methochloride
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
(-)-Bicuculline methochloride
😃Good
Catalog No. T12044Alias l-Bicuculline methochlorideCas No. 53552-05-9
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $160 | 35 days | |
| 10 mg | $288 | 35 days | |
| 25 mg | $630 | 35 days | |
| 50 mg | $987 | 35 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | (-)-Bicuculline methochloride is a potent antagonist of GABAA receptor. |
| In vivo | In rat ,(-)-Bicuculline methochloride (0.6 nmol/rat) weaken the antiallodynic effect of Neurotropin[2]. |
| Alias | l-Bicuculline methochloride |
| Molecular Weight | 417.84 |
| Formula | C21H20ClNO6 |
| Cas No. | 53552-05-9 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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